click below
click below
Normal Size Small Size show me how
BetaBlockers
Fundamentals II
Question | Answer |
---|---|
Atenolol | selective, lowest lipid solubility, 12-14 hr 1/2 life, oral administration, #1 drug for HTN, angina, hyperthyroidism |
Esmolol | selective, 10 min 1/2 life, IV administration, antiarrythmis |
Metoprolol | selective, high lipid solubility, 3-6 hr 1/2 life, oral administration, some MSA, used for HTN, angina, hyperthyroidism |
Celiprolol | selective, used for HTN and angina |
Naldolol | non-selective, 24 hr 1/2 life, oral administration, used for HTN & angina |
Propranolol | non-selective, highest lipid solubility, highest plasma binding, 3-6 hr 1/2 life, OH propranolol is active metabolite, oral & IV administration, highest MSA (mouth gets numb), used for HTN, angina, & antiarrythmic |
Pindolol | non-selective, 3-6 hr 1/2 life, oral administration, highest ISA, some MSA, used for HTN & angina |
Timolol | non-selective, 3-6 hr 1/2 life, oral administration, #1 drug for glaucoma, used for HTN, angina, & hyperthyroidism |
Labetalol | non-selective, but selective alpha1 blocker, 3-6 hr 1/2 life, oral administration, HTN & angina |