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pharam
Term | Definition |
---|---|
atropine | ACH receptor inhibitor |
endrophonium | short term Ach esterase inhibitor |
neostigmine | medium term Ach esterase inhibitor |
physostigmine | medium term Ach esterase inhibitor |
phyrimadostigmine | medium term Ach esterase inhibitor |
isoflurophate | long term Ach esterase inhibitor |
palidoxamine | reverse the inhibition of isoflurophate |
Tacrine | Prototypical AChE inhibitor for AD |
Donepezil | reversible acetylcholinesterase inhibitor |
Rivastigmine | Parkinson disease |
Galantamine | Competitive, reversible AChE inhibitor |
succinylcholine | depolarizing agent |
d-tubocuraine | non depolarizing agent main poision blocks the NMm RECEPTOR |
curare | paralyzes affect the ach release, but it does not affect when they are taken in orally because the stomach breaks them down and releases it. |
Fasiculation | muscle twitching |
plasma acetylcholinesterase ;butyrylcholinesterase | to prolong the activity of break the Succinylcholine |
suxamethonium or succylcholine | muscle relaxant during anaesthesia |
sarin, tabun, soman | they are all gases used as nerve agents |
Hemicholinium | Competitive inhibitor of choline uptake (not taken up itself |
Vesamicol | Inhibition of packaging of acetylcholine into vesicles |
Triethylcholine | Inhibits choline uptake, taken up and acetylated to acetyltriethylcholine. Stored as a false transmitter (i.e. normal vesicular release) |
Muscarinic cholinomimetics | resemble the effects of parasympathetic stimulation |